Moetsi oa Cabazixel oa boleng bo phahameng ba cabazitaxel

Tlhaloso e Khutšoanyane:

Carbataxel ke ntho ea lik'hemik'hale e sebelisoang ho etsa litlhare tse thibelang mofetše.Carbataxel ke phofo e tšoeu kapa e tšoeu e batlang e sa qhibilihe ka metsing, empa e qhibiliha ka ethanol.Mokhoa oa eona oa ho thibela mofetše le litšobotsi li tšoana le docetaxel, 'me ke ea sehlopha sa lithethefatsi tse khahlanong le microtubule.Ka ho kopanya le tubulin, ho khothalletsa ho bokana lona ka microtubules, ka nako e tšoanang ho ka thibela tsena e bokana microtubule disassembly, hore tsitsisa microtubules, ka tsela eo inhibiting mitosis seleng, 'me interphase cell function (interphasecellularfunctions).


Lintlha tsa Sehlahisoa

Li-tag tsa Sehlahisoa

Litaba tsa Sehlahisoa

Lebitso:Cabazitaxel

Nomoro ea CAS:183133-96-2

Foromo ea lik'hemik'hale:C45H57NO14

Litlhaloso:99%

Mmala:phofo e tshweu kapa e bosweu

Mohloli:Semi-synthesized le 10-DAB

Mofuta:APIs

Karolo le melemo ea cabataxel

1.anti-cancer effect: carbamazel e na le phello e matla e khahlanong le kankere, e ka thibela ka katleho ho hōla le ho ata ha lisele tsa tumor, ho etsa hore apoptosis ea lisele tsa tumor e be teng.Ha ho bapisoa le paclitaxel ea tlhaho, carbataxel e na le ts'ebetso e phahameng ea anti-cancer le spectrum e pharaletseng ea anti-cancer.

2.tšireletseho: Cabataxel ka mokhoa oa ho qapa le ho etsa lihlahisoa, tsepamisa maikutlo ho ntlafatsa tšireletso ea lihlahisoa le mamello.Ka ho fetola le ho ntlafatsa sebopeho sa lik'hemik'hale tsa paclitaxel, liketsahalo tsa litla-morao le liketso tse mpe li ile tsa fokotseha.

Litšobotsi tsa 3.pharmacokinetic: carbamazel e na le litšobotsi tse molemo tsa pharmacokinetic, e le hore e ka kenngoa hantle le ho ajoa 'meleng, e le ho ntlafatsa phello ea phekolo.

4.applicability: carbataxel e ka sebelisoa ho phekola mefuta e sa tšoaneng ea kankere, ho akarelletsa le kankere ea matšoafo, kankere ea matsoele, kankere ea mahe a bomme, kankere ea mala, joalo-joalo. Ho sebetsa ha eona le ho sireletseha ho 'nile ha netefatsoa ka hohle-hohle.

5.Tšehetso ea saense: Cabataxel e itšetlehile ka lipatlisiso tsa morao-rao tsa saense le tsoelo-pele ea theknoloji, ka tšehetso e tšepahalang ea saense.

Litšebeletso tsa Rōna

1.Lihlahisoa:Fana ka lihlahisoa tsa limela tsa boleng bo holimo, tse hloekileng haholo, lisebelisoa tse tala tsa meriana, le li-intermediate tsa meriana.

2.Litšebeletso tsa tekheniki:Li-extracts tse ikhethileng tse nang le litlhaloso tse khethehileng ho latela litlhoko tsa bareki.

Hande fektheri

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