Fektheri e phahameng ea 10-DAB Semi-synthetic Paclitaxel GMP

Tlhaloso e Khutšoanyane:

10-DAB semi-synthetic paclitaxel ke setlhare se thibelang hlahala se sebetsang hantle haholo ebile se bolokehile, se nang le tebello e pharalletseng ea ts'ebeliso.Ke semi-synthesized semi-synthesized ho tloha paclitaxel ea tlhaho le metsoako ea maiketsetso, e bolokang ts'ebetso e ntle ea anti-tumor ea paclitaxel, ha e ntse e ntlafatsa katleho ea tlhahiso le bohloeki ba lithethefatsi.


Lintlha tsa Sehlahisoa

Li-tag tsa Sehlahisoa

Litaba tsa Sehlahisoa

Lebitso:10-DAT Semi-synthetic Paclitaxel

Nomoro ea CAS:33069-62-4

Foromo ea lik'hemik'hale:C47H51NO14

Litlhaloso:99%-102%

Mmala:phofo e tshweu kapa e batlile e tshweu

Mohloli:Taxus yunnanensis, Taxus chinensis

Mofuta:APIs

Mokhoa oa ho tseba le bophelo ba sethala

Mokhoa oa ho lemoha:HPLC

Ho nepahala:3 lilemo

Nako ea tlhahlobo hape:Likhoeli tse 36

Bokhoni ba letsoho:600-800kg / selemo

Phello

10-DAB semi-synthetic paclitaxel e na le mesebetsi e mengata kalafong ea tumor.Ke sethethefatsi se sebetsang hantle se khahlanong le hlahala, se ka thibelang karohano le ho ata ha lisele tsa hlahala, ho khothaletsa apoptosis, le ho eketsa kutlo ea lisele tsa hlahala ho radiotherapy le chemotherapy.Ho phaella moo, sethethefatsi sena se na le bioavailability e ntle 'me se ka kenngoa ka ho feletseng ke lisele tsa hlahala, ho ntlafatsa phello ea phekolo.E boetse e na le nako e telele ea halofo ea bophelo, e ka fokotsang tšitiso ea tsamaiso khafetsa.Ha ho bapisoa le lihlahisoa tse ling tse tšoanang, 10-DAB semi-synthetic paclitaxel e na le litla-morao tse tlase tsa chefo 'me e loketse haholoanyane kalafo ea nako e telele.Setlhare sena se ka boela sa fetola ts'ebetso ea pharmacological ea paclitaxel ka ho fetola sebopeho sa eona, kahoo e fana ka menyetla e mengata ea nts'etsopele ea lithethefatsi.

Litšebeletso tsa Rōna

1.Lihlahisoa:Fana ka lihlahisoa tsa limela tsa boleng bo holimo, tse hloekileng haholo, lisebelisoa tse tala tsa meriana, le li-intermediate tsa meriana.

2.Litšebeletso tsa tekheniki:Li-extracts tse ikhethileng tse nang le litlhaloso tse khethehileng ho latela litlhoko tsa bareki.

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