Cabazitaxel Cas 183133-96-2 Moetsi oa Cabazitaxil

Tlhaloso e Khutšoanyane:

Carbataxel ke ntho ea lik'hemik'hale e sebelisoang ho etsa litlhare tse thibelang mofetše.Carbataxel ke phofo e tšoeu kapa e tšoeu e batlang e sa qhibilihe ka metsing, empa e qhibiliha ka ethanol.Mokhoa oa eona oa ho thibela mofetše le litšobotsi li tšoana le docetaxel, 'me ke ea sehlopha sa lithethefatsi tse khahlanong le microtubule.Ka ho kopanya le tubulin, ho khothalletsa ho bokana lona ka microtubules, ka nako e tšoanang ho ka thibela tsena e bokana microtubule disassembly, hore tsitsisa microtubules, ka tsela eo inhibiting mitosis seleng, 'me interphase cell function (interphasecellularfunctions).


Lintlha tsa Sehlahisoa

Li-tag tsa Sehlahisoa

Litaba tsa Sehlahisoa

Lebitso:Cabazitaxel

Nomoro ea CAS:183133-96-2

Foromo ea lik'hemik'hale:C45H57NO14

Litlhaloso:99%

Mmala:phofo e tshweu kapa e bosweu

Mohloli:Semi-synthesized le 10-DAB

Mofuta:APIs

Phello

Carbataxel ke derivative ea taxane e sebetsang e le microtubule inhibitor, e tlamang tubulin le ho khothaletsa kopano ea eona ho li-microtubules, ha e ntse e thibela ho arohana ha li-microtubules tsena tse bokaneng le ho tsitsisa li-microtubules.Thibelo ena e fella ka ho senyeha ha li-microtubules le ho khaotsa ho arohana ha lisele, kahoo ho emisa potoloho ea lisele le ho thibela ho ata ha hlahala.Ka hona, carbataxel e sebelisoa haholo-holo bakeng sa ho lokisa lithethefatsi tse khahlanong le mofetše, e na le phello e ntle ea ho thibela kankere, 'me e ka sebelisoa ho phekola mafu a sa tšoaneng a baktheria.Ka ho khetheha, carbataxel e 'nile ea sebelisoa haholo ho phekola tšoelesa ea senya, matsoele, mahe a bomme, matšoafo, le mafu a mang a mangata a kankere, hammoho le tšoaetso ea baktheria, ho akarelletsa le sinusitis, bronchitis, pneumonia, tšoaetso ea moroto, tšoaetso ea mahlo, tšoaetso ea letlalo le otitis media.

Litšebeletso tsa Rōna

1.Lihlahisoa:Fana ka lihlahisoa tsa limela tsa boleng bo holimo, tse hloekileng haholo, lisebelisoa tse tala tsa meriana, le li-intermediate tsa meriana.

2.Litšebeletso tsa tekheniki:Li-extracts tse ikhethileng tse nang le litlhaloso tse khethehileng ho latela litlhoko tsa bareki.

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