Lekhasi la amora DNJ lekhasi la mulberry le ntša sehlahisoa sa bophelo bo botle

Tlhaloso e Khutšoanyane:

Lekhasi la Mulberry DNJ ke alkaloid ea tlhaho, eo lebitso la eona la Sechaena e leng 1-deoxynojirimycin.Ke enzyme e matla ea glucose metabolizing (mohlala, α- Glycosidase) inhibitor e ka liehisang ts'ebetso ea ho senyeha ha polysaccharide, ea fokotsa boleng ba tlhōrō ea tsoekere ea mali ka mor'a lijo le ho tsitsisa tsoekere e potlakileng ea mali;Ke ea "inhibitory factor" har'a lintlha tse 'ne tse laolang tsoekere ea alfa.


Lintlha tsa Sehlahisoa

Li-tag tsa Sehlahisoa

Litaba tsa Sehlahisoa

Lekhasi la Mulberry DNJ ke alkaloid ea tlhaho, eo lebitso la eona la Sechaena e leng 1-deoxynojirimycin.Ke enzyme e matla ea glucose metabolizing (mohlala, α- Glycosidase) inhibitor e ka liehisang ts'ebetso ea ho senyeha ha polysaccharide, ea fokotsa boleng ba tlhōrō ea tsoekere ea mali ka mor'a lijo le ho tsitsisa tsoekere e potlakileng ea mali;Ke ea "inhibitory factor" har'a lintlha tse 'ne tse laolang tsoekere ea alfa.
1、 Phello ea lekhasi la amora DNJ
1. Tsela e meraro ea ho fokotsa tsoekere ea mali
Joalo ka inhibitor e matla ea li-enzyme tse ntlafatsang tsoekere (mohlala, α- Glucosidase, hexokinase, glucuronidase le glycogen phosphatase, joalo-joalo), DNJ e ka liehisa ts'ebetso ea pholiso ea polysaccharide haholo, ea fokotsa boleng ba tlhōrō ea tsoekere ea mali ea postprandial le ho tsitsisa tsoekere ea mali e potlakileng.Ho feta moo, DNJ e na le phello ea insulin sensitization ho ntlafatsa ho hanyetsa insulin.
2. Fokotsa tsoekere ea mali ea postprandial.
α- Glucosidase e ajoa haholo ka maleng a motho mme e bapala karolo ea bohlokoa ho bola ha lik'habohaedreite.Ba ikarabella bakeng sa ho senyeha ha li-oligosaccharides tse kang oligosaccharides lijong ka monosaccharides, tse kang glucose.Glucose ena e kena 'meleng ka lerako la mala, e leng se bakang ho phahama ho hoholo ha tsoekere ea mali.DNJ ke ea tlhaho ebile e matla α-Glucosidase inhibitors e tlamang ka tlholisano mala a manyane α- Kamano ea glucosidase e phahame ho feta ea oligosaccharides joalo ka sucrose le maltose α-Glucosidase e na le kamano e matla mme e fokotsa li-oligosaccharides le α-glucosidability. , e le ho thibela ho bola ha fructose ho tsoekere, 'me palo e kholo ea tsoekere e ke ke ea kenngoa le ho romeloa mala a maholo.Ka lebaka la phello ea DNJ, tsoekere e nyane e kena maling, kahoo tsoekere ea mali e lokela ho bolokoa e le maemong a phetseng hantle.
3. Glucose ea mali e tsitsitseng.
DNJ e na le ts'ebetso ea inhibitory ea glycogen phosphorylase, e ka liehisang ho senyeha ha sebete sa glycogen hore e be tsoekere, e le ho tsitsisa tsoekere ea mali e potlakileng.Glucose e "feteletseng" 'meleng oa motho e bolokiloe ka har'a sebete ka sebopeho sa glycogen.Glycogen e ka aroloa hore e be tsoekere tlas'a ts'ebetso ea glycogen phosphorylase 'me ea lokolloa maling ho finyella litlhoko tsa mesifa le mesebetsi e meng ea litho.Glycogen ke o mong oa mehloli e meholo ea matla bakeng sa boikoetliso ba 'mele.Ka phetoho e tšoanang lipakeng tsa glycogen le glucose, tsoekere ea mali ea batho ba tloaelehileng e leka-lekaneng.Ho bakuli ba nang le lefu la tsoekere, ka lebaka la ho se sebetse hantle ha metabolism ea tsoekere, glycogen e ngata haholo e tla oela ho glucose, e leng se bakang keketseho e sa tloaelehang ea tsoekere ea mali e potlakileng.DNJ e ka thibela tšebetso ea glycogen phosphorylase le ho thibela keketseho ea tsoekere ea mali e bakoang ke ho bola ho feteletseng ha glycogen ho ba tsoekere, e le ho tsitsisa tsoekere ea mali e potlakileng.
4. Ntlafatsa ho hanyetsa insulin.
DNJ e ka ntlafatsa matšoao a ho hanyetsa insulin ka ho lokisa lipid metabolism, ho liehisa tlhahiso ea tsoekere le ho matlafatsa insulin.Ho hanyetsa insulin ho bolela mabaka a fapaneng (haholo-holo a kenyeletsang liphatsa tsa lefutso le botenya), tse fokotsang katleho ea insulin e khothalletsang ho amoheloa le ho sebelisoa ha tsoekere, 'me' mele o fana ka insulin e ngata ka mokhoa o khotsofatsang.Ho hanyetsa insulin ho hlahisa hyperinsulinemia ho boloka botsitso ba tsoekere ea mali 'meleng.Haeba 'mele oa motho o le maemong a ho hanyetsa insulin nako e telele, o tla eketsa moroalo oa manyeme haholo.E ka etsa hore manyeme a hlahise ho se sebetse hantle ha insulin, ebe joale a fetoha lefu la tsoekere.DNJ e ka ntlafatsa matšoao a ho hanyetsa insulin ka ho boloka tsoekere ea mali e phetse hantle, ho lokisa lipid metabolism le ho eketsa kutloisiso ea insulin.
2、 Masimo a kopo ea lekhasi la amora DNJ
Letlapa la 'Mulberry lekhasi la DNJ le thathamisitsoe e le phello e thusang ea hypoglycemic mme e sebelisoa haholo lijong tsa bophelo bo botle.

Lihlahisoa tsa lihlahisoa

BOEMO BA KHOEBO
Lebitso la Sehlahiswa Lekhasi la Mulberry DNJ
CAS 19130-96-2
Foromo ea Lik'hemik'hale C6H13NO4
Branta Hlee
Mmohlahisi YUnnan Hande Bio-Tech Co., Ltd.
Ckantle Kunming,China
E thehiloe 1993
 BASIC TSEBISO
Litlhaloso tse tšoanang (2r, 3r, 4r,5s) -2-hydroxymethyl-3,4,5-trihydroxypiperidine;5-piperidinetriol,2-(hydroxymethyl)-,(2r-(2alpha,3beta,4alpha,5beta)) -4;bay-h5595;moranolin;moranoline;

(+)-1-DEOXYNOJIRIMYCIN;1-DEOXYNOJIRIMYCIN;(2R,3R,4R,5S)-2-(HYDROXYMETHYL)-3,4,5-PIPERIDINETRIOL

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Polelo ea sehlahisoa sa Hande

1.Lihlahisoa tsohle tse rekisoang ke k'hamphani ke lisebelisoa tse tala tse felileng.Lihlahisoa li lebisitsoe haholo ho bahlahisi ba nang le mangolo a tlhahiso, 'me lisebelisoa tse tala ha se lihlahisoa tsa ho qetela.
2.Theko e ka bang teng le lits'ebetso tse amehang kenyelletsong kaofela li tsoa libukeng tse hatisitsoeng.Batho ka bomong ha ba khothaletse tšebeliso e tobileng, 'me ho reka ka bomong ho haneloa.
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